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Tocris Bioscience™ MSC 2032964A
Potent and selective ASK1 inhibitor; orally bioavailable
Marca: Tocris Bioscience™ 5641/10
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Descripción
MSC 2032964A is a potent and selective ASK1 inhibitor (IC50 = 93 nM). Selective for ASK1 over a panel of 210 kinases. Blocks LPS-induced ASK1 and p38 phosphorylation in cultured mouse astrocytes. Suppresses neuroinflammation in a mouse EAE model. Orally bioavailable and brain penetrant.Especificaciones
N-[5-(Cyclopropylamino)-7-(trifluoromethyl)[1,2,4]triazolo[1,5-a]pyridin-2-yl]-3-pyridinecarboxamide | |
1124381-43-6 | |
10 mg |