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STEMCELL Technologies Fasudil (Dihydrochloride)
RHO/ROCK pathway inhibitor; Inhibits ROCK2
Marca: STEMCELL Technologies 73664

Descripción
- Fasudil (also known as HA-1077) is a potent inhibitor of Rho-associated coiled-coil containing protein kinase 2 (ROCK2; IC50 = 1.9 μM)
- Additionally, it inhibits protein kinase C-related kinase 2 (PRK2), mitogen- and stress-activated protein kinase (MSK1), and mitogen-activated protein kinase-activated protein kinase 1b (MAPKAP-K1b) with IC50 values of 4, 5, and 15 μM, respectively (Davies et al.) This product is supplied as the dihydrochloride salt of the molecule
Especificaciones
203911-27-7 | |
100 mg | |
≥98% |
HA-1077 | |
C14H17N3O2S · 2HCl |
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